Target Classes > GPCRs > Ortholog

Ortholog GPCR Assay List

DiscoveRx offers a comprehensive range of non-human ortholog GPCR assays to facilitate counterscreening and SAR evaluation of compounds identified in a primary screen using a human GPCR target. The DiscoveRx Services platform leverages this menu of GPCR assays for all screening and profiling services.

 

  • Overview of Available Readout

Arrestin


Browse Available Ortholog GPCR Targets

Listed below are the assays currently available for screening and profiling.  Assays may be sorted by column name. Contact us if you don't see your target of interest in the list below as additional catalog assays may be available for screening and profiling as a custom service.
Family ▲Target GeneCommon NameSpeciesG protein couplingAccession NumberArrestin
5-Hydroxytryptamine mHTR2Am5HT2AMouseGi/GoNM_172812X
5-Hydroxytryptamine mHTR2Cm5HT2CMouseGi/GoAF498983X
AcetylcholinerCHRM4rM4RatGs & Gi/GoNM_000741X
AdenosinemADORA2BmA2BMouseGs NM_007413X
AdenosinemADORA3mA3MouseGi/GoNM_009631.3X
AnaphylatoxinmC5AR1mC5ARMouseGi/GoNM_007577.3X
ApelinmAGTRL1mAPJMouseGi/GoNM_011784.2X
CannabinoidmCNR1mCB1MouseGi/GoNM_007726X
CannabinoidmCNR2mCB2MouseGi/GoNM_009924X
ChemokinemCCR1mCC1MouseGi/GoNM_009912X
ChemokinemCCR10mCCR10MouseGi/GoAY429103X
ChemokinemCCR2mCCR2MouseGi/GoNM_009915.2X
ChemokinemCCR3mCCR3MouseGi/GoNM_009914X
ChemokinemCCR4mCCR4MouseGi/GoNM_006619X
ChemokinemCCR5mCCR5MouseGi/GoNM_009917X
ChemokinemCCR6mCCR6MouseGi/GoNM_009835.3X
ChemokinemCCR7mCCR7MouseGi/GoNM_007719.2X
ChemokinemCCR8mCCR8MouseGi/GoNM_007720.2X
ChemokinemCMKLR1mCMKLR1MouseGi/GoNM_008153.2X
ChemokinemCXCR2mCXCR2MouseGi/GoNM_009909X
ChemokinemCXCR3mCXCR3MouseGi/GoNM_009910X
ChemokinemCXCR4mCXCR4MouseGi/GoXM_001478244.1X
ChemokinemCXCR5mCXCR5MouseGi/GoNM_007551X
ChemokinemCXCR6mCXCR6MouseGi/GoNM_030712X
ChemokinemCXCR7mCXCR7MouseNoneNM_007722X
Chemokine mCCR9mCCR9MouseGi/GoNM_007713.5X
Class A OrphanmGPR1mGPR1MouseUnknownNM_146250X
Class A OrphanmGPR120mGPR120MouseUnknownNM_181748X
CorticotropinmCRHR1mCRF1MouseGsNM_007762X
DopaminemDRD5mDRD5MouseGsNM_013503.2X
DopaminerDRD2LrD2LRatGi/GoNM_012547.1X
DopaminerDRD2SrD2SRatGi/GoNM_016574.3X
DopaminerDRD5rD5RatGsNM_000798.3X
EndothelinmEDNRAmETAMouseGqNM_010332.2X
EndothelinmEDNRBmETBMouseGi/Go & GsNM_007904.3X
Formylpeptide mFPR1mFPR1MouseGqNM_013521.2X
GalaninmGALR2mGALR2MouseGi/GoNM_010254.4X
GhrelinmGHSR1aghrelinMouseGqNM_177330X
GlucagonmGCGRglucagonMouseGsNM_008101.2X
GlucagonmGIPRmGIPMouseGsNM_001080815.1X
GlucagonmGLP1RmGLP-1MouseGsNM_021332X
LeukotrienemLTB4RmBLT1MouseGi/Go & GqNM_008519.2X
LysophospholipidcEDG5cS1P2CanineGsXM_542076.2X
LysophospholipidmEDG1mS1P1MouseGi/GoNM_007901X
LysophospholipidmEDG5mS1P2MouseGsNM_010333.4X
LysophospholipidmEDG6mS1P4MouseGqNM_010102.2X
LysophospholipidrEDG5rS1P2RatGsNM_017192.2X
LysophospholipidsEDG5sS1P2SimianGsXM_001100481.1X
Melanin-concentrating hormonemMCHR1MCH1MouseGi/GoNM_145132X
Neuropeptide YmNPY1RY1MouseGi/GoNM_010934.4X
Neuropeptide YmNPY2RNPY2RMouseGi/Go & GqNM_008731.3X
Neuropeptide YmPPYR1Y4MouseGi/GoNM_008919.4X
OpioidmOPRD1δ (murine)MouseGi/GoNM_013622.3X
OpioidmOPRK1κ (murine)MouseGi/GoNM_011011X
OpioidmOPRM1μ (murine)MouseGi/GoNM_001039652X
OpioidrOPRM1μRatGi/GoNM_013071X
OrexinmHCRTR1mOX1MouseGqAY062030X
P2YmP2RY12mP2Y12MouseGi/GoNM_027571.3X
P2YmP2RY6P2Y6MouseGqNM_183168.1X
Platelet-activating factor mPTAFRmPAFMouseGi/Go & GqNM_001081211.1X
ProkineticinrPROKR1rPROKR1RatGs & Gq X
ProkineticinrPROKR2rPKR2RatGsNM_138978X
ProstanoidmCRTH2mDP2MouseGi/GoNM_009962.2X
ProstanoidrCRTH2rGPR44RatGi/GoNM_001012070.1X
SomatostatinmSSTR2mSST2MouseGi/GoNM_001042606.1X
SomatostatinmSSTR5mSRIF1BMouseGi/GoNM_011425.2X
UrotensinmUTR2mUTMouseGqNM_145440X
Vasopressin and OxytocinmOXTR1mOTMouseGqNM_001081147.1X
VIP and PACAPmADCYAP1R1mPAC1MouseGs & GqNM_001025372.1X
VIP and PACAPmVIPR1mVPAC1MouseGsNM_011703.4X