Explore our Assay Panels
View complete list of assays and available panels
DiscoveRx services offer a comprehensive portfolio of cell-based and biochemical assay formats against a broad range of target classes. View available assays and assay panels below. Don't see the assay you need?
Contact us if you don't see your target of interest in our list below as additional catalog items may be available for screening and profiling as a custom service.
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Browse Complete Target List
Listed below are the assays currently available for screening and profiling. Assays may be sorted by column name.
Contact us if you don't see your target of interest in list below as additional catalog assays may be available for screening and profiling as a custom service.
| Target Class ▲ | Family/Group | Target Gene | Common Name | Species |
| GPCR | VIP and PACAP | ADCYAP1R1 | PAC1 | Human |
| GPCR | Adenosine | ADORA1 | A1 | Human |
| GPCR | Adenosine | ADORA2A | A2A | Human |
| GPCR | Adenosine | ADORA2B | A2B | Human |
| GPCR | Adenosine | ADORA3 | A3 | Human |
| GPCR | Adrenergic | ADRA1A | α1A-adrenoreceptor | Human |
| GPCR | Adrenergic | ADRA1B | α1B-adrenoreceptor | Human |
| GPCR | Adrenergic | ADRA2A | α2A-adrenoreceptor | Human |
| GPCR | Adrenergic | ADRA2B | α2B-adrenoreceptor | Human |
| GPCR | Adrenergic | ADRA2C | α2C-adrenoreceptor | Human |
| GPCR | Adrenergic | ADRB1 | β1-adrenoreceptor | Human |
| GPCR | Adrenergic | ADRB2 | β2-adrenoreceptor | Human |
| GPCR | Adrenergic | ADRB3 | β3-adrenoreceptor | Human |
| GPCR | Angiotensin | AGTR1 | AT1 | Human |
| GPCR | Apelin | AGTRL1 | APJ | Human |
| GPCR | Vasopressin and Oxytocin | AVPR1A | V1A | Human |
| GPCR | Vasopressin and Oxytocin | AVPR1B | V1B | Human |
| GPCR | Vasopressin and Oxytocin | AVPR2 | V2 | Human |
| GPCR | Class B Orphan | BAI1 | BAI1 | Human |
| GPCR | Class B Orphan | BAI2 | BAI2 | Human |
| GPCR | Class B Orphan | BAI3 | BAI3 | Human |
| GPCR | Bradykinin | BDKRB1 | B1 | Human |
| GPCR | Bradykinin | BDKRB2 | B2 | Human |
| GPCR | Bombesin | BRS3 | BB3 | Human |
| GPCR | Anaphylatoxin | C3AR1 | C3A | Human |
| GPCR | Anaphylatoxin | C5AR1 | C5A | Human |
| GPCR | Anaphylatoxin | C5L2 | C5L2 | Human |
| GPCR | Calcitonin | CALCR | CT | Human |
| GPCR | Calcitonin | CALCR + RAMP1 | AMY1 | Human |
| GPCR | Calcitonin | CALCR + RAMP2 | AMY2 | Human |
| GPCR | Calcitonin | CALCR + RAMP3 | AMY3 | Human |
| GPCR | Calcitonin | CALCRL + RAMP1 | CGRP | Human |
| GPCR | Calcitonin | CALCRL + RAMP2 | AM1 | Human |
| GPCR | Calcitonin | CALCRL + RAMP3 | AM2 | Human |
| GPCR | Calcium sensing | CASR | CaS | Human |
| GPCR | Cholecystokinin | CCKAR | CCK1 | Human |
| GPCR | Cholecystokinin | CCKBR | CCK2 | Human |
| GPCR | Chemokine | CCR1 | CCR1 | Human |
| GPCR | Chemokine | CCR10 | CCR10 | Human |
| GPCR | Chemokine | CCR2 | CCR2 | Human |
| GPCR | Chemokine | CCR3 | CCR3 | Human |
| GPCR | Chemokine | CCR4 | CCR4 | Human |
| GPCR | Chemokine | CCR5 | CCR5 | Human |
| GPCR | Chemokine | CCR6 | CCR6 | Human |
| GPCR | Chemokine | CCR7 | CCR7 | Human |
| GPCR | Chemokine | CCR8 | CCR8 | Human |
| GPCR | Chemokine | CCR9 | CCR9 | Human |
| GPCR | Class A Orphan | CCRL2 | CCRL2 | Human |
| GPCR | Lysophospholipid | cEDG5 | cS1P2 | Canine |
| GPCR | Acetylcholine | CHRM1 | M1 | Human |
| GPCR | Acetylcholine | CHRM2 | M2 | Human |
| GPCR | Acetylcholine | CHRM3 | M3 | Human |
| GPCR | Acetylcholine | CHRM4 | M4 | Human |
| GPCR | Acetylcholine | CHRM5 | M5 | Human |
| GPCR | Chemokine | CMKLR1 | CMKLR1 | Human |
| GPCR | Cannabinoid | CNR1 | CB1 | Human |
| GPCR | Cannabinoid | CNR2 | CB2 | Human |
| GPCR | Corticotropin | CRHR1 | CRF1 | Human |
| GPCR | Corticotropin | CRHR2 | CRF2 | Human |
| GPCR | Prostanoid | CRTH2 | DP2 | Human |
| GPCR | Chemokine | CX3CR1 | CX3CR1 | Human |
| GPCR | Chemokine | CXCR1 | CXCR1 | Human |
| GPCR | Chemokine | CXCR2 | CXCR2 | Human |
| GPCR | Chemokine | CXCR3 | CXCR3 | Human |
| GPCR | Chemokine | CXCR4 | CXCR4 | Human |
| GPCR | Chemokine | CXCR5 | CXCR5 | Human |
| GPCR | Chemokine | CXCR6 | CXCR6 | Human |
| GPCR | Chemokine | CXCR7 | CXCR7 | Human |
| GPCR | Leukotriene | CYSLTR2 | CYSLT2 | Human |
| GPCR | Non-signalling 7TM chemokine-binding proteins | DARC | FY | Human |
| GPCR | Dopamine | DRD1 | D1 | Human |
| GPCR | Dopamine | DRD2L | D2L | Human |
| GPCR | Dopamine | DRD2S | D2S | Human |
| GPCR | Dopamine | DRD3 | D3 | Human |
| GPCR | Dopamine | DRD4 | D4 | Human |
| GPCR | Dopamine | DRD5 | D5 | Human |
| GPCR | Class A Orphan | EBI2 | GPR183 | Human |
| GPCR | Lysophospholipid | EDG1 | S1P1 | Human |
| GPCR | Lysophospholipid | EDG2 | LPA1 | Human |
| GPCR | Lysophospholipid | EDG3 | S1P3 | Human |
| GPCR | Lysophospholipid | EDG4 | LPA2 | Human |
| GPCR | Lysophospholipid | EDG5 | S1P2 | Human |
| GPCR | Lysophospholipid | EDG6 | S1P4 | Human |
| GPCR | Lysophospholipid | EDG7 | LPA3 | Human |
| GPCR | Lysophospholipid | EDG8 | S1P5 | Human |
| GPCR | Endothelin | EDNRA | ETA | Human |
| GPCR | Endothelin | EDNRB | ETB | Human |
| GPCR | Protease activated | F2R | PAR1 | Human |
| GPCR | Protease activated | F2RL1 | PAR2 | Human |
| GPCR | Protease activated | F2RL3 | PAR4 | Human |
| GPCR | Free Fatty Acid | FFAR1 | FFA1 | Human |
| GPCR | Free Fatty Acid | FFAR2 | GPR43 | Human |
| GPCR | Free Fatty Acid | FFAR3 | GPR41 | Human |
| GPCR | Formylpeptide | FPR1 | FPR1 | Human |
| GPCR | Formylpeptide | FPRL1 | FPR2/ALX | Human |
| GPCR | Glycoprotein hormone receptor | FSHR | FSHR | Human |
| GPCR | GABAB | GABBR1 | GABB1 | Human |
| GPCR | Galanin | GALR1 | GALR1 | Human |
| GPCR | Galanin | GALR2 | GALR2 | Human |
| GPCR | Glucagon | GCGR | glucagon | Human |
| GPCR | Glucagon | GHRHR | GHRH | Human |
| GPCR | Ghrelin | GHSR1a | ghrelin | Human |
| GPCR | Class A Orphan | GHSR1b | GHSR1b | Human |
| GPCR | Glucagon | GIPR | GIP | Human |
| GPCR | Glucagon | GLP1R | GLP-1 | Human |
| GPCR | Glucagon | GLP2R | GLP-2 | Human |
| GPCR | Gonadotropin-releasing hormone | GNRHR | GnRH | Human |
| GPCR | Bile acid | GPBAR1 | GPBA | Human |
| GPCR | Class A Orphan | GPR1 | GPR1 | Human |
| GPCR | Class A Orphan | GPR101 | GPR101 | Human |
| GPCR | Peptide P518 receptor | GPR103 | QRFPR | Human |
| GPCR | Other 7TM proteins | GPR107 | GPR107 | Human |
| GPCR | Hydroxycarboxylic acid | GPR109A | HCA2 | Human |
| GPCR | Hydroxycarboxylic acid | GPR109B | HCA3 | Human |
| GPCR | Class A Orphan | GPR119 | GPR119 | Human |
| GPCR | Class A Orphan | GPR12 | GPR12 | Human |
| GPCR | Class A Orphan | GPR120 | GPR120 | Human |
| GPCR | Class B Orphan | GPR123 | GPR123 | Human |
| GPCR | Class A Orphan | GPR132 | GPR132 | Human |
| GPCR | Class A Orphan | GPR135 | GPR135 | Human |
| GPCR | Other 7TM proteins | GPR137 | TM7SF1 | Human |
| GPCR | Class A Orphan | GPR139 | GPR139 | Human |
| GPCR | Class A Orphan | GPR141 | GPR141 | Human |
| GPCR | Class A Orphan | GPR142 | GPR142 | Human |
| GPCR | Other 7TM proteins | GPR143 | GPR143 | Human |
| GPCR | Class A Orphan | GPR146 | GPR146 | Human |
| GPCR | Class A Orphan | GPR148 | GPR148 | Human |
| GPCR | Class A Orphan | GPR149 | GPR149 | Human |
| GPCR | Class A Orphan | GPR15 | GPR15 | Human |
| GPCR | Class A Orphan | GPR150 | GPR150 | Human |
| GPCR | Class A Orphan | GPR151 | GPR151 | Human |
| GPCR | Class A Orphan | GPR152 | GPR152 | Human |
| GPCR | Class B Orphan | GPR157 | GPR157 | Human |
| GPCR | Class A Orphan | GPR161 | GPR161 | Human |
| GPCR | Class A Orphan | GPR162 | GPR162 | Human |
| GPCR | Class A Orphan | GPR17 | GPR17 | Human |
| GPCR | Class A Orphan | GPR171 | GPR171 | Human |
| GPCR | Class A Orphan | GPR173 | GPR173 | Human |
| GPCR | Class A Orphan | GPR176 | GPR176 | Human |
| GPCR | Class A Orphan | GPR18 | GPR18 | Human |
| GPCR | Class A Orphan | GPR182 | GPR182 | Human |
| GPCR | Class A Orphan | GPR20 | GPR20 | Human |
| GPCR | Class A Orphan | GPR23 | LPA4 | Human |
| GPCR | Class A Orphan | GPR25 | GPR25 | Human |
| GPCR | Class A Orphan | GPR26 | GPR26 | Human |
| GPCR | Class A Orphan | GPR27 | GPR27 | Human |
| GPCR | Class A Orphan | GPR3 | GPR3 | Human |
| GPCR | Estrogen (G protein coupled) receptor | GPR30 | GPER | Human |
| GPCR | Class A Orphan | GPR31 | GPR31 | Human |
| GPCR | Class A Orphan | GPR32 | GPR32 | Human |
| GPCR | Class A Orphan | GPR35 | GPR35 | Human |
| GPCR | Class A Orphan | GPR37 | EDNRBL | Human |
| GPCR | Class A Orphan | GPR37L1 | GPR37L1 | Human |
| GPCR | Class A Orphan | GPR39 | GPR39 | Human |
| GPCR | Class A Orphan | GPR4 | GPR4 | Human |
| GPCR | Class A Orphan | GPR45 | GPR45 | Human |
| GPCR | Class A Orphan | GPR50 | GPR50 | Human |
| GPCR | Class A Orphan | GPR52 | GPR52 | Human |
| GPCR | Class A Orphan | GPR55 | GPR55 | Human |
| GPCR | Class A Orphan | GPR6 | GPR6 | Human |
| GPCR | Class A Orphan | GPR61 | GPR61 | Human |
| GPCR | Class A Orphan | GPR65 | GPR65 | Human |
| GPCR | Class A Orphan | GPR75 | GPR75 | Human |
| GPCR | Class A Orphan | GPR78 | GPR78 | Human |
| GPCR | Class A Orphan | GPR79 | GPR79 | Human |
| GPCR | Hydroxycarboxylic acid | GPR81 | HCA1 | Human |
| GPCR | Class A Orphan | GPR83 | GPR83 | Human |
| GPCR | Class A Orphan | GPR84 | GPR84 | Human |
| GPCR | Class A Orphan | GPR85 | GPR85 | Human |
| GPCR | Class A Orphan | GPR88 | GPR88 | Human |
| GPCR | Class A Orphan | GPR91 | SUCNR1 | Human |
| GPCR | Class A Orphan | GPR92 | GPR92 | Human |
| GPCR | Class B Orphan | GPR97 | GPR97 | Human |
| GPCR | Glutamate | GRM1 | mGlu1 | Human |
| GPCR | Glutamate | GRM2 | mGlu2 | Human |
| GPCR | Glutamate | GRM3 | MGlu3 | Human |
| GPCR | Glutamate | GRM4 | mGlu4 | Human |
| GPCR | Glutamate | GRM6 | mGlu6 | Human |
| GPCR | Bombesin | GRPR | BB2 | Human |
| GPCR | Orexin | HCRTR1 | OX1 | Human |
| GPCR | Orexin | HCRTR2 | OX2 | Human |
| GPCR | Histamine | HRH1 | H1 | Human |
| GPCR | Histamine | HRH2 | H2 | Human |
| GPCR | Histamine | HRH3 | H3 | Human |
| GPCR | Histamine | HRH4 | H4 | Human |
| GPCR | 5-Hydroxytryptamine | HTR1A | 5HT1A | Human |
| GPCR | 5-Hydroxytryptamine | HTR1B | 5HT1B | Human |
| GPCR | 5-Hydroxytryptamine | HTR1E | 5HT1E | Human |
| GPCR | 5-Hydroxytryptamine | HTR1F | 5HT1F | Human |
| GPCR | 5-Hydroxytryptamine | HTR2A | 5HT2A | Human |
| GPCR | 5-Hydroxytryptamine | HTR2B | 5HT2B | Human |
| GPCR | 5-Hydroxytryptamine | HTR2C | 5HT2C | Human |
| GPCR | 5-Hydroxytryptamine | HTR5A | 5HT5A | Human |
| GPCR | 5-Hydroxytryptamine | HTR7A | 5HT7A | Human |
| GPCR | 5-Hydroxytryptamine | HTR7B | 5HT7B | Human |
| GPCR | 5-Hydroxytryptamine | HTR7D | 5HT7D | Human |
| GPCR | Kisspeptin receptor | KISS1R | kisspeptin | Human |
| GPCR | Class A Orphan | LGR4 | LGR4 | Human |
| GPCR | Class A Orphan | LGR5 | LGR5 | Human |
| GPCR | Class A Orphan | LGR6 | LGR6 | Human |
| GPCR | Glycoprotein hormone receptor | LHCGR | LH | Human |
| GPCR | Leukotriene | LTB4R | BLT1 | Human |
| GPCR | VIP and PACAP | mADCYAP1R1 | mPAC1 | Mouse |
| GPCR | Adenosine | mADORA2B | mA2B | Mouse |
| GPCR | Adenosine | mADORA3 | mA3 | Mouse |
| GPCR | Apelin | mAGTRL1 | mAPJ | Mouse |
| GPCR | Melanocortin | MC1R | MC1 | Human |
| GPCR | Melanocortin | MC3R | MC3 | Human |
| GPCR | Melanocortin | MC4R | MC4 | Human |
| GPCR | Anaphylatoxin | mC5AR1 | mC5AR | Mouse |
| GPCR | Melanocortin | MC5R | MC5 | Human |
| GPCR | Chemokine | mCCR1 | mCC1 | Mouse |
| GPCR | Chemokine | mCCR10 | mCCR10 | Mouse |
| GPCR | Chemokine | mCCR2 | mCCR2 | Mouse |
| GPCR | Chemokine | mCCR3 | mCCR3 | Mouse |
| GPCR | Chemokine | mCCR4 | mCCR4 | Mouse |
| GPCR | Chemokine | mCCR5 | mCCR5 | Mouse |
| GPCR | Chemokine | mCCR6 | mCCR6 | Mouse |
| GPCR | Chemokine | mCCR7 | mCCR7 | Mouse |
| GPCR | Chemokine | mCCR8 | mCCR8 | Mouse |
| GPCR | Chemokine | mCCR9 | mCCR9 | Mouse |
| GPCR | Melanin-concentrating hormone | MCHR1 | MCH1 | Human |
| GPCR | Melanin-concentrating hormone | MCHR2 | MCH2 | Human |
| GPCR | Chemokine | mCMKLR1 | mCMKLR1 | Mouse |
| GPCR | Cannabinoid | mCNR1 | mCB1 | Mouse |
| GPCR | Cannabinoid | mCNR2 | mCB2 | Mouse |
| GPCR | Corticotropin | mCRHR1 | mCRF1 | Mouse |
| GPCR | Prostanoid | mCRTH2 | mDP2 | Mouse |
| GPCR | Chemokine | mCXCR2 | mCXCR2 | Mouse |
| GPCR | Chemokine | mCXCR3 | mCXCR3 | Mouse |
| GPCR | Chemokine | mCXCR4 | mCXCR4 | Mouse |
| GPCR | Chemokine | mCXCR5 | mCXCR5 | Mouse |
| GPCR | Chemokine | mCXCR6 | mCXCR6 | Mouse |
| GPCR | Chemokine | mCXCR7 | mCXCR7 | Mouse |
| GPCR | Dopamine | mDRD5 | mDRD5 | Mouse |
| GPCR | Lysophospholipid | mEDG1 | mS1P1 | Mouse |
| GPCR | Lysophospholipid | mEDG5 | mS1P2 | Mouse |
| GPCR | Lysophospholipid | mEDG6 | mS1P4 | Mouse |
| GPCR | Endothelin | mEDNRA | mETA | Mouse |
| GPCR | Endothelin | mEDNRB | mETB | Mouse |
| GPCR | Formylpeptide | mFPR1 | mFPR1 | Mouse |
| GPCR | Galanin | mGALR2 | mGALR2 | Mouse |
| GPCR | Glucagon | mGCGR | glucagon | Mouse |
| GPCR | Ghrelin | mGHSR1a | ghrelin | Mouse |
| GPCR | Glucagon | mGIPR | mGIP | Mouse |
| GPCR | Glucagon | mGLP1R | mGLP-1 | Mouse |
| GPCR | Class A Orphan | mGPR1 | mGPR1 | Mouse |
| GPCR | Class A Orphan | mGPR120 | mGPR120 | Mouse |
| GPCR | Orexin | mHCRTR1 | mOX1 | Mouse |
| GPCR | 5-Hydroxytryptamine | mHTR2A | m5HT2A | Mouse |
| GPCR | 5-Hydroxytryptamine | mHTR2C | m5HT2C | Mouse |
| GPCR | Motilin | MLNR | motilin | Human |
| GPCR | Leukotriene | mLTB4R | mBLT1 | Mouse |
| GPCR | Melanin-concentrating hormone | mMCHR1 | MCH1 | Mouse |
| GPCR | Neuropeptide Y | mNPY1R | Y1 | Mouse |
| GPCR | Neuropeptide Y | mNPY2R | NPY2R | Mouse |
| GPCR | Opioid | mOPRD1 | δ (murine) | Mouse |
| GPCR | Opioid | mOPRK1 | κ (murine) | Mouse |
| GPCR | Opioid | mOPRM1 | μ (murine) | Mouse |
| GPCR | Vasopressin and Oxytocin | mOXTR1 | mOT | Mouse |
| GPCR | P2Y | mP2RY12 | mP2Y12 | Mouse |
| GPCR | P2Y | mP2RY6 | P2Y6 | Mouse |
| GPCR | Neuropeptide Y | mPPYR1 | Y4 | Mouse |
| GPCR | Platelet-activating factor | mPTAFR | mPAF | Mouse |
| GPCR | Class A Orphan | MRGPRD | MRGPRD | Human |
| GPCR | Class A Orphan | MRGPRE | MRGPRE | Human |
| GPCR | Class A Orphan | MRGPRF | MRGPRF | Human |
| GPCR | Class A Orphan | MRGPRX1 | MRGPRX1 | Human |
| GPCR | Class A Orphan | MRGPRX2 | MRGX2 | Human |
| GPCR | Class A Orphan | MRGPRX4 | MRGPRX4 | Human |
| GPCR | Somatostatin | mSSTR2 | mSST2 | Mouse |
| GPCR | Somatostatin | mSSTR5 | mSRIF1B | Mouse |
| GPCR | Melatonin | MTNR1A | MT1 | Human |
| GPCR | Melatonin | MTNR1B | MT2 | Human |
| GPCR | Urotensin | mUTR2 | mUT | Mouse |
| GPCR | VIP and PACAP | mVIPR1 | mVPAC1 | Mouse |
| GPCR | Neuromedin U | NMU1R | NMU1 | Human |
| GPCR | Neuropeptide B & W | NPBWR1 | NPBW1 | Human |
| GPCR | Neuropeptide B & W | NPBWR2 | NPBW2 | Human |
| GPCR | Neuropeptide F | NPFFR1 | NPFF1 | Human |
| GPCR | Neuropeptide F | NPFFR2 | NPFF2 | Human |
| GPCR | Neuropeptide S | NPSR1B | NPS receptor | Human |
| GPCR | Neuropeptide Y | NPY1R | Y1 | Human |
| GPCR | Neuropeptide Y | NPY2R | Y2 | Human |
| GPCR | Neurotensin | NTSR1 | NTS1 | Human |
| GPCR | Class A Orphan | OPN5 | OPN5 | Human |
| GPCR | Opioid | OPRD1 | δ | Human |
| GPCR | Opioid | OPRK1 | κ | Human |
| GPCR | Opioid | OPRL1 | NOP | Human |
| GPCR | Opioid | OPRM1 | μ | Human |
| GPCR | Leukotriene | OXER1 | OXE | Human |
| GPCR | Class A Orphan | OXGR1 | OXGR1 | Human |
| GPCR | Vasopressin and Oxytocin | OXTR | OT | Human |
| GPCR | P2Y | P2RY1 | P2RY1 | Human |
| GPCR | P2Y | P2RY11 | P2Y11 | Human |
| GPCR | P2Y | P2RY12 | P2Y12 | Human |
| GPCR | P2Y | P2RY2 | P2Y2 | Human |
| GPCR | P2Y | P2RY4 | P2Y4 | Human |
| GPCR | P2Y | P2RY6 | P2Y6 | Human |
| GPCR | Class A Orphan | P2RY8 | P2RY8 | Human |
| GPCR | Neuropeptide Y | PPYR1 | Y4 | Human |
| GPCR | Prolactin releasing peptide receptor | PRLHR | PRRP | Human |
| GPCR | Prokineticin | PROKR1 | PKR1 | Human |
| GPCR | Prokineticin | PROKR2 | PKR2 | Human |
| GPCR | Platelet-activating factor | PTAFR | PAF | Human |
| GPCR | Prostanoid | PTGDR | DP1 | Human |
| GPCR | Prostanoid | PTGER1 | EP1 | Human |
| GPCR | Prostanoid | PTGER2 | EP2 | Human |
| GPCR | Prostanoid | PTGER3 | EP3 | Human |
| GPCR | Prostanoid | PTGER4 | EP4 | Human |
| GPCR | Prostanoid | PTGFR | FP | Human |
| GPCR | Prostanoid | PTGIR | IP1 | Human |
| GPCR | Parathyroid | PTHR1 | PTH1 | Human |
| GPCR | Parathyroid | PTHR2 | PTH2 | Human |
| GPCR | Acetylcholine | rCHRM4 | rM4 | Rat |
| GPCR | Prostanoid | rCRTH2 | rGPR44 | Rat |
| GPCR | Dopamine | rDRD2L | rD2L | Rat |
| GPCR | Dopamine | rDRD2S | rD2S | Rat |
| GPCR | Dopamine | rDRD5 | rD5 | Rat |
| GPCR | Lysophospholipid | rEDG5 | rS1P2 | Rat |
| GPCR | Opioid | rOPRM1 | μ | Rat |
| GPCR | Prokineticin | rPROKR1 | rPROKR1 | Rat |
| GPCR | Prokineticin | rPROKR2 | rPKR2 | Rat |
| GPCR | Relaxin | RXFP1 | RXFP1 | Human |
| GPCR | Relaxin | RXFP3 | RXFP3 | Human |
| GPCR | Relaxin | RXFP4 | RXFP4 | Human |
| GPCR | Glucagon | SCTR | secretin | Human |
| GPCR | Lysophospholipid | sEDG5 | sS1P2 | Simian |
| GPCR | Somatostatin | SSTR1 | SST1 | Human |
| GPCR | Somatostatin | SSTR2 | SST2 | Human |
| GPCR | Somatostatin | SSTR3 | SST3 | Human |
| GPCR | Somatostatin | SSTR4 | SST4 | Human |
| GPCR | Somatostatin | SSTR5 | SST5 | Human |
| GPCR | Class A Orphan | TAAR5 | TAAR5 | Human |
| GPCR | Tachykinin | TACR1 | NK1 | Human |
| GPCR | Tachykinin | TACR2 | NK2 | Human |
| GPCR | Tachykinin | TACR3 | NK3 | Human |
| GPCR | Prostanoid | TBXA2R | TP | Human |
| GPCR | TRH | TRHR | TRH1 | Human |
| GPCR | Glycoprotein hormone receptor | TSHR(L) | TSH | Human |
| GPCR | Urotensin | UTR2 | UT | Human |
| GPCR | VIP and PACAP | VIPR1 | VPAC1 | Human |
| GPCR | VIP and PACAP | VIPR2 | VPAC2 | Human |
| GPCR | Chemokine | XCR1 | XCR1 | Human |
| KINASE | RTK | AXL | AXL | Human |
| KINASE | RTK | c-KIT | c-KIT | Human |
| KINASE | RTK | c-MET | C-MET | Human |
| KINASE | CTK | CSF3R | | Human |
| KINASE | CTK | CSF3R-JAK1 | | Human |
| KINASE | RTK | EphA5 | EphA5 | Human |
| KINASE | RTK | EphA7 | EphA7 | Human |
| KINASE | RTK | EphB2 | EphB2 | Human |
| KINASE | RTK | EphB3 | EphB3 | Human |
| KINASE | RTK | EphB4 | EphB4 | Human |
| KINASE | RTK | ErbB1 | EGFR | Human |
| KINASE | RTK | ErbB2 | HER2 | Human |
| KINASE | RTK | ErbB2/ErbB3 | HER2/HER3 | Human |
| KINASE | RTK | ErbB4 | HER4 | Human |
| KINASE | CTK | GHR | | Human |
| KINASE | CTK | GHR-JAK1 | | Human |
| KINASE | CTK | GHR-JAK2 | | Human |
| KINASE | RTK | IGF1R | IGF1R | Human |
| KINASE | RTK | INSR | INSR | Human |
| KINASE | RTK | PDGFRA | PDGFRa | Human |
| KINASE | RTK | PDGFRB | PDGFRb | Human |
| KINASE | CTK | PRLR | PRLR | Human |
| KINASE | CTK | PRLR-JAK1 | | Human |
| KINASE | CTK | PRLR-JAK2 | | Human |
| KINASE | CTK | SYK | | Human |
| KINASE | RTK | TrkA | NTRK1 | Human |
| KINASE | RTK | TrkA-p75 | TrkA-p75 | Human |
| KINASE | RTK | TrkB | NTRK2 | Human |
| KINASE | RTK | TrkB-p75 | TrkB-p75 | Human |
| KINASE | RTK | TrkC | NTRK3 | Human |
| KINASE | RTK | TrkC-p75 | TrkC-p75 | Human |
| KINASE | CTK | TYK2 | | Human |
| NHR | NHR | AR | | Human |
| NHR | NHR | ERRα | | Human |
| NHR | NHR | ERα | | Human |
| NHR | NHR | FXR | | Human |
| NHR | NHR | GR | GR | Human |
| NHR | NHR | LXRb-NCoR1 | | Human |
| NHR | NHR | LXRα | LXRα | Human |
| NHR | NHR | LXRβ | LXRβ | Human |
| NHR | NHR | MR | MR | Human |
| NHR | NHR | PPARα | | Human |
| NHR | NHR | PPARγ | | Human |
| NHR | NHR | PPARδ | | Human |
| NHR | NHR | PRα | | Human |
| NHR | NHR | PRβ | | Human |
| NHR | NHR | RARα | | Human |
| NHR | NHR | RARβ | | Human |
| NHR | NHR | RORg | | Human |
| NHR | NHR | RXRα | | Human |
| NHR | NHR | RXRγ | | Human |
| NHR | NHR | THRα | | Human |
| NHR | NHR | THRβ | | Human |
| Pathway | Pathway | ADCY2 | adenylate cyclase 2 | Human |
| Pathway | Pathway | CDC25A | | Human |
| Pathway | Pathway | FOXO3 | forkhead box O3 | Human |
| Pathway | Pathway | GSK3β | β-Catenin Translocation | Human |
| Pathway | Pathway | IkB | IkB | Human |
| Pathway | Pathway | Keap1 NRF2 | Keap1&Nrf2 | Human |
| Pathway | Pathway | NPR1 | NPR1 | Human |
| Pathway | Pathway | P53 | | Human |
| Pathway | Pathway | PDK/AKT | FOXO3 Translocation | Human |
| Pathway | Pathway | PI3 | FOXO3 Translocation | Human |
| Pathway | Pathway | SREBP2 | SREBF2 | Human |
| Pathway | Pathway | TNFα | IkB Degradation | Human |
| Pathway | Pathway | Wnt3 | β-Catenin Translocation | Human |
| Pathway | Pathway | XBP1 | XBP1 | Human |